Abstract
The synthesis of a suitably protected sugar amino acid (δ-glyco-amino acid) as a building block to be incorporated into the peptide chain (N-terminus) of bioactive peptide analogues is described. Its efficient coupling reactions with pilot amino acids as well as dipeptides have been accomplished by standard peptide chemistry.
Original language | English |
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Pages (from-to) | 845-852 |
Number of pages | 8 |
Journal | Synthesis |
Issue number | 6 |
DOIs | |
Publication status | Published - 16 Mar 2007 |
Keywords
- δ-glyco-amino acid
- Carbohydrates
- Glycopeptides
- Glycosylation
- Radiolabelling